A novel method for the facile synthesis of depsipeptides

Chaim Gilon; Yakir Klausner; Alfred Hassner

doi:10.1016/S0040-4039(01)95531-5

A novel method for the facile synthesis of depsipeptides

Chaim Gilon^*
, Yakir Klausner
, Alfred Hassner

^*Corresponding author for this work

Institute of Chemistry

Research output: Contribution to journal › Article › peer-review

68 Scopus citations

Abstract

A one pot, high yield synthesis of depsipeptides is described involving room temperature condensation of hindered substrates (N-Boc amino acids and benzyl α-hydroxy esters) in the presence of DCC and a dialkylaminopyridine. In this manner previously inaccessible depsipeptides were prepared.

Original language	English
Pages (from-to)	3811-3814
Number of pages	4
Journal	Tetrahedron Letters
Volume	20
Issue number	40
DOIs	https://doi.org/10.1016/S0040-4039(01)95531-5
State	Published - 1979

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10.1016/S0040-4039(01)95531-5

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title = "A novel method for the facile synthesis of depsipeptides",

abstract = "A one pot, high yield synthesis of depsipeptides is described involving room temperature condensation of hindered substrates (N-Boc amino acids and benzyl α-hydroxy esters) in the presence of DCC and a dialkylaminopyridine. In this manner previously inaccessible depsipeptides were prepared.",

author = "Chaim Gilon and Yakir Klausner and Alfred Hassner",

year = "1979",

doi = "10.1016/S0040-4039(01)95531-5",

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T1 - A novel method for the facile synthesis of depsipeptides

AU - Gilon, Chaim

AU - Klausner, Yakir

AU - Hassner, Alfred

PY - 1979

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N2 - A one pot, high yield synthesis of depsipeptides is described involving room temperature condensation of hindered substrates (N-Boc amino acids and benzyl α-hydroxy esters) in the presence of DCC and a dialkylaminopyridine. In this manner previously inaccessible depsipeptides were prepared.

AB - A one pot, high yield synthesis of depsipeptides is described involving room temperature condensation of hindered substrates (N-Boc amino acids and benzyl α-hydroxy esters) in the presence of DCC and a dialkylaminopyridine. In this manner previously inaccessible depsipeptides were prepared.

UR - https://www.scopus.com/pages/publications/49249151511

U2 - 10.1016/S0040-4039(01)95531-5

DO - 10.1016/S0040-4039(01)95531-5

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AN - SCOPUS:49249151511

SN - 0040-4039

VL - 20

SP - 3811

EP - 3814

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 40

ER -

A novel method for the facile synthesis of depsipeptides

Abstract

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