Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands

Fabrizio Fierro, Lior Peri, Harald Hübner, Alina Tabor-Schkade, Lukas Waterloo, Stefan Löber, Tara Pfeiffer, Dorothee Weikert, Tamir Dingjan, Eitan Margulis, Peter Gmeiner*, Masha Y. Niv*

*Corresponding author for this work

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Keyphrases

Chemistry

Biochemistry, Genetics and Molecular Biology

Pharmacology, Toxicology and Pharmaceutical Science